By Emeritus Professor David Black

Journal articles

Kuppusamy R; Willcox M; Black DSC; Kumar N, 2019, 'Short cationic peptidomimetic antimicrobials', Antibiotics, 8, pp. 44, http://dx.doi.org/10.3390/antibiotics8020044

Hong KKC; Ho KKK; Bhadbhade M; Ball GE; Black DS; Kumar N, 2019, 'The Mosaic of Rottlerin: The Sequel', Journal of Natural Products, 82, pp. 1190 - 1199, http://dx.doi.org/10.1021/acs.jnatprod.8b00917

Almohaywi B; Yu TT; Iskander G; Chan DSH; Ho KKK; Rice S; Black DSC; Griffith R; Kumar N, 2019, 'Dihydropyrrolones as bacterial quorum sensing inhibitors', Bioorganic and Medicinal Chemistry Letters, 29, pp. 1054 - 1059, http://dx.doi.org/10.1016/j.bmcl.2019.03.004

Dobrowolski JC; Nguyen DHT; Fraser BH; Bhadbhade M; Black DSC; Kumar N, 2019, 'A General Synthesis of 7-Phenyl-7,13-dihydro-8 H -benzo[6,7]azepino[3,2- c ]quinolin-8-ones', Synlett, 30, pp. 567 - 572, http://dx.doi.org/10.1055/s-0037-1612106

Dobrowolski JC; Nguyen DHT; Fraser BH; Bhadbhade M; Black DSC; Kumar N, 2019, 'A General Synthesis of Benzoazepinoindoles-A New Class of Heterocycles', Synlett, 30, pp. 2081 - 2085, http://dx.doi.org/10.1055/s-0039-1690700

Wenholz DS; Bhadbhade M; Kandemir H; Ho J; Kumar N; Black DS, 2019, 'Substituent effects in solid-state assembly of activated benzotriazoles', CrystEngComm, 21, pp. 835 - 842, http://dx.doi.org/10.1039/c8ce01757c

Jumina J; Wenholz DS; Kumar N; Black DS, 2019, 'Synthesis of a Variety of Activated Pyrrolo[3,2,1- ij ]quinolines', Synthesis (Germany), 51, pp. 1989 - 1994, http://dx.doi.org/10.1055/s-0037-1612280

Yee EMH; Cirillo G; Brandl MB; Black DSC; Vittorio O; Kumar N, 2019, 'Synthesis of dextran–phenoxodiol and evaluation of its physical stability and biological activity', Frontiers in Bioengineering and Biotechnology, 7, http://dx.doi.org/10.3389/fbioe.2019.00183

Qu J; Bhadbhade M; Kumar N; Black DSC, 2018, 'Unusual formation of novel highly substituted N-(3-indolyl)-imidazoles', Tetrahedron, 74, pp. 7438 - 7441, http://dx.doi.org/10.1016/j.tet.2018.11.007

Beyer RL; Kandemir H; Bhadbhade M; Sengul IF; Leu CW; Wenholz D; Kumar N; Black DSC, 2018, 'Synthesis of dipyrrolo[2,3-a:1′,2′,3′-fg]acridin-12(1H)-ones', Tetrahedron Letters, 59, pp. 4483 - 4486, http://dx.doi.org/10.1016/j.tetlet.2018.11.011

Taunk A; Chen R; Iskander G; Ho KKK; Black DSC; Willcox MDP; Kumar N, 2018, 'Dual-Action Biomaterial Surfaces with Quorum Sensing Inhibitor and Nitric Oxide to Reduce Bacterial Colonization', ACS Biomaterials Science and Engineering, 4, pp. 4174 - 4182, http://dx.doi.org/10.1021/acsbiomaterials.8b00816

Almohaywi B; Iskander G; Yu TT; Bhadbhade M; Black DSC; Kumar N, 2018, 'Copper-mediated Chan-Evans-Lam N-arylation of 5-methylene-4-aryl-1,5-dihydro-2H-pyrrol-2-one derivatives', Tetrahedron Letters, 59, pp. 811 - 814, http://dx.doi.org/10.1016/j.tetlet.2018.01.039

Biswas NN; Iskander GM; Mielczarek M; Yu TT; Black DSC; Kumar N, 2018, 'Alkyne-Substituted Fimbrolide Analogues as Novel Bacterial Quorum-Sensing Inhibitors', Australian Journal of Chemistry, 71, pp. 708 - 715, http://dx.doi.org/10.1071/CH18194

Almohaywi B; Taunk A; Wenholz DS; Nizalapur S; Biswas NN; Ho KKK; Rice SA; Iskander G; Black DSC; Griffith R; Kumar N, 2018, 'Design and synthesis of lactams derived from mucochloric and mucobromic acids as pseudomonas aeruginosa quorum sensing inhibitors', Molecules, 23, http://dx.doi.org/10.3390/molecules23051106

Kuppusamy R; Yasir M; Berry T; Cranfield CG; Nizalapur S; Yee E; Kimyon O; Taunk A; Ho KKK; Cornell B; Manefield M; Willcox M; Black DSC; Kumar N, 2018, 'Design and synthesis of short amphiphilic cationic peptidomimetics based on biphenyl backbone as antibacterial agents', European Journal of Medicinal Chemistry, 143, pp. 1702 - 1722, http://dx.doi.org/10.1016/j.ejmech.2017.10.066

Aldilla VR; Martin AD; Nizalapur S; Marjo CE; Rich AM; Ho KKK; Ittner LM; Black DSC; Thordarson P; Kumar N, 2018, 'Glyoxylamide-based self-assembly hydrogels for sustained ciprofloxacin delivery', Journal of Materials Chemistry B, 6, pp. 6089 - 6098, http://dx.doi.org/10.1039/C8TB01290C

Kuppusamy R; Yasir M; Yee E; Willcox M; Black DSC; Kumar N, 2018, 'Guanidine functionalized anthranilamides as effective antibacterials with biofilm disruption activity', Organic and Biomolecular Chemistry, 16, pp. 5871 - 5888, http://dx.doi.org/10.1039/c8ob01699b

Suryanti V; Bhadbhade M; Black DSC; Kumar N, 2017, 'N-acetylglyoxylic amide bearing a nitrophenyl group as anion receptors: NMR and X-ray investigations on anion binding and selectivity', Journal of Molecular Structure, 1146, pp. 571 - 576, http://dx.doi.org/10.1016/j.molstruc.2017.05.133

Dobrowolski JC; Fraser BH; Bhadbhade M; Black DS; Kumar N, 2017, 'Efficient Access to Chromeno[4,3- b ]quinolines Related to Dependensin', Synlett, 28, pp. 1979 - 1983, http://dx.doi.org/10.1055/s-0036-1589087

将樹 北; 修 大; 薫 山; 英夫 木; 大輔 上; Black DS, 2017, '30 有毒哺乳動物カモノハシ由来の神経毒に関する生物有機化学的研究(口頭発表の部)', , pp. 175 - 180, http://dx.doi.org/10.24496/tennenyuki.52.0_175

Deodhar M; Black DS; Kumar N, 2017, 'P-479 SYNTHESIS OF DIMERIC FLAVONOIDS RELATED TO DEPENDENSIN AND ITS ANALOGUES', , pp. _p - 479_, http://dx.doi.org/10.24496/intnaturalprod.2006.0__p-479_

Yee EMH; Hook JM; Bhadbhade MM; Vittorio O; Kuchel RP; Brandl MB; Tilley RD; Black DSC; Kumar N, 2017, 'Preparation, characterization and in vitro biological evaluation of (1:2) phenoxodiol-β-cyclodextrin complex', Carbohydrate Polymers, 165, pp. 444 - 454, http://dx.doi.org/10.1016/j.carbpol.2017.02.081

Yu TT; Nizalapur S; Ho KKK; Yee E; Berry T; Cranfield CG; Willcox M; Black DSC; Kumar N, 2017, 'Design, Synthesis and Biological Evaluation of N-Sulfonylphenyl glyoxamide-Based Antimicrobial Peptide Mimics as Novel Antimicrobial Agents', ChemistrySelect, 2, pp. 3452 - 3461, http://dx.doi.org/10.1002/slct.201700336

Nizalapur S; Kimyon O; Yee E; Ho K; Berry T; Manefield M; Cranfield CG; Willcox M; Black DSC; Kumar N, 2017, 'Amphipathic guanidine-embedded glyoxamide-based peptidomimetics as novel antibacterial agents and biofilm disruptors', Organic and Biomolecular Chemistry, 15, pp. 2033 - 2051, http://dx.doi.org/10.1039/C7OB00053G

Aldilla VR; Nizalapur S; Martin A; Marjo CE; Rich A; Yee E; Suwannakot P; Black DS; Thordarson P; Kumar N, 2017, 'Design, synthesis, and characterisation of glyoxylamide-based short peptides as self-assembled gels', New Journal of Chemistry, 41, pp. 13462 - 13471, http://dx.doi.org/10.1039/c7nj02248d

Dobrowolski JC; Somphol K; Santoso M; Duong H; Gardner CR; Kumar N; Black DSC, 2017, 'Methanal extrusion in ipso-substitution reactions of hydroxymethylindoles', Australian Journal of Chemistry, 70, pp. 1188 - 1195, http://dx.doi.org/10.1071/CH17257

Wenholz DS; Zeng M; Ma C; Mielczarek M; Yang X; Bhadbhade M; Black DSC; Lewis PJ; Griffith R; Kumar N, 2017, 'Small molecule inhibitors of bacterial transcription complex formation', Bioorganic and Medicinal Chemistry Letters, 27, pp. 4302 - 4308, http://dx.doi.org/10.1016/j.bmcl.2017.08.036

Nizalapur S; Kimyon O; Yee E; Bhadbhade MM; Manefield M; Willcox M; Black DS; Kumar N, 2017, 'Synthesis and biological evaluation of novel acyclic and cyclic glyoxamide based derivatives as bacterial quorum sensing and biofilm inhibitors', Organic and Biomolecular Chemistry, 15, pp. 5743 - 5755, http://dx.doi.org/10.1039/c7ob01011g

Biswas NN; Yu TT; Kimyon Ö; Nizalapur S; Gardner CR; Manefield M; Griffith R; Black DSC; Kumar N, 2017, 'Synthesis of antimicrobial glucosamides as bacterial quorum sensing mechanism inhibitors', Bioorganic and Medicinal Chemistry, 25, pp. 1183 - 1194, http://dx.doi.org/10.1016/j.bmc.2016.12.024

Kandemir H; Sengul IF; Kumar N; Black DSC, 2017, 'Synthesis of imine and amine-linked macrocycles containing tris-indoles', Australian Journal of Chemistry, 70, pp. 1196 - 1201, http://dx.doi.org/10.1071/CH17264

Yee EMH; Brandl MB; Black DSC; Vittorio O; Kumar N, 2017, 'Synthesis of isoflavene-thiosemicarbazone hybrids and evaluation of their anti-tumor activity', Bioorganic and Medicinal Chemistry Letters, 27, pp. 2454 - 2458, http://dx.doi.org/10.1016/j.bmcl.2017.04.002

Bingul M; Tan O; Gardner CR; Sutton SK; Arndt GM; Marshall GM; Cheung BB; Kumar N; Black DSC; Arndt G, 2016, 'Synthesis, characterization and anti-cancer activity of hydrazide derivatives incorporating a quinoline moiety', Molecules, 21, pp. 916, http://dx.doi.org/10.3390/molecules21070916

Kandemir H; Sengul IF; Kumar N; Black DSC, 2016, 'Synthesis of a 7-(aminomethyl)indole and related bis-indole derivatives', Arkivoc, 2016, pp. 288 - 295, http://dx.doi.org/10.3998/ark.5550190.p009.587

Nizalapur S; Ho KKK; Kimyon Ö; Yee E; Berry T; Manefield M; Cranfield CG; Willcox M; Black DSC; Kumar N, 2016, 'Synthesis and biological evaluation of N-naphthoyl-phenylglyoxamide-based small molecular antimicrobial peptide mimics as novel antimicrobial agents and biofilm inhibitors', Organic and Biomolecular Chemistry, 14, pp. 3623 - 3637, http://dx.doi.org/10.1039/c6ob00298f

Thach O; Mielczarek M; Ma C; Kutty SK; Yang X; Black DSC; Griffith R; Lewis PJ; Kumar N, 2016, 'From indole to pyrrole, furan, thiophene and pyridine: Search for novel small molecule inhibitors of bacterial transcription initiation complex formation', Bioorganic and Medicinal Chemistry, 24, pp. 1171 - 1182, http://dx.doi.org/10.1016/j.bmc.2016.01.040

Biswas NN; Kutty SK; Iskander GM; Mielczarek M; Bhadbhade MM; Gardner CR; Black DSC; Kumar N, 2016, 'Synthesis of brominated novel N-heterocycles: New scaffolds for antimicrobial discovery', Tetrahedron, 72, pp. 539 - 546, http://dx.doi.org/10.1016/j.tet.2015.12.018

Bingul M; Kumar N; Black DS, 2016, 'Synthesis and reactions of new 2-hydroxymethyldimethoxyindoles', Tetrahedron, 72, pp. 234 - 239, http://dx.doi.org/10.1016/j.tet.2015.11.038

Dobrowolski JC; Katen A; Fraser BH; Bhadbhade M; Black DSC; Kumar N, 2016, 'A general and efficient synthesis of 5,6-dihydrodibenzo[b,h][1,6]naphthyridine derivatives', Tetrahedron Letters, 57, pp. 5442 - 5445, http://dx.doi.org/10.1016/j.tetlet.2016.10.067

Nizalapur S; Kimyon Ö; Biswas NN; Gardner CR; Griffith R; Rice SA; Manefield M; Willcox M; Black DSC; Kumar N, 2016, 'Design, synthesis and evaluation of N-aryl-glyoxamide derivatives as structurally novel bacterial quorum sensing inhibitors', Organic and Biomolecular Chemistry, 14, pp. 680 - 693, http://dx.doi.org/10.1039/c5ob01973g

Kandemir H; Sengul IF; Gardner CR; Werry EL; Barron ML; Kassiou M; Kumar N; Black DSC, 2016, 'Synthesis of 7,7′-linked-bis-indoles via 7-tryptamines', Heterocycles, 93, pp. 333 - 346, http://dx.doi.org/10.3987/COM-15-S(T)55

Biswas NN; Kutty SK; Iskander GM; Mielczarek M; Bhadbhade MM; Gardner CR; Black DS; Kumar N, 2016, 'ChemInform Abstract: Synthesis of Brominated Novel N‐Heterocycles: New Scaffolds for Antimicrobial Discovery.', ChemInform, 47, http://dx.doi.org/10.1002/chin.201620030

Goh WK; Gardner CR; Chandra Sekhar KVG; Biswas NN; Nizalapur S; Rice SA; Willcox M; Black DS; Kumar N, 2015, 'Synthesis, quorum sensing inhibition and docking studies of 1,5-dihydropyrrol-2-ones', Bioorganic and Medicinal Chemistry, 23, pp. 7366 - 7377, http://dx.doi.org/10.1016/j.bmc.2015.10.025

Mielczarek M; Bhadbhade M; Chen R; Kumar N; Black DSC, 2015, 'Bromination of 2,7′-bi-indolyls and quinazolin-7-ones', Tetrahedron, 71, pp. 8925 - 8942, http://dx.doi.org/10.1016/j.tet.2015.09.064

Chen Y; Cass SL; Kutty SK; Yee EMH; Chan DSH; Gardner CR; Vittorio O; Pasquier E; Black DSC; Kumar N, 2015, 'Synthesis, biological evaluation and structure-activity relationship studies of isoflavene based Mannich bases with potent anti-cancer activity', Bioorganic and Medicinal Chemistry Letters, 25, pp. 5377 - 5383, http://dx.doi.org/10.1016/j.bmcl.2015.09.027

Hong KKC; Ball GE; Black DS; Kumar N, 2015, 'The Mosaic of Rottlerin', Journal of Organic Chemistry, 80, pp. 10668 - 10674, http://dx.doi.org/10.1021/acs.joc.5b01827

Kutty SK; Barraud N; Ho KKK; Iskander GM; Griffith R; Rice SA; Bhadbhade M; Willcox MDP; Black DS; Kumar N, 2015, 'Hybrids of acylated homoserine lactone and nitric oxide donors as inhibitors of quorum sensing and virulence factors in Pseudomonas aeruginosa', Organic and Biomolecular Chemistry, 13, pp. 9850 - 9861, http://dx.doi.org/10.1039/c5ob01373a

Mielczarek M; Thomas RV; Ma C; Kandemir H; Yang X; Bhadbhade M; Black DS; Griffith R; Lewis PJ; Kumar N, 2015, 'Synthesis and biological activity of novel mono-indole and mono-benzofuran inhibitors of bacterial transcription initiation complex formation', Bioorganic and Medicinal Chemistry, 23, pp. 1763 - 1775, http://dx.doi.org/10.1016/j.bmc.2015.02.037

Iskander G; Wood K; Eiffe E; Yee EMH; Black DSC; Kumar N, 2015, 'Ritter reactions of isoflavanols: A facile route to 4-amidoisoflavans', Tetrahedron Letters, 56, pp. 1941 - 1943, http://dx.doi.org/10.1016/j.tetlet.2015.02.072

Biswas NN; Kutty SK; Barraud N; Iskander GM; Griffith R; Rice SA; Willcox M; Black DS; Kumar N, 2015, 'Indole-based novel small molecules for the modulation of bacterial signalling pathways', Organic and Biomolecular Chemistry, 13, pp. 925 - 937, http://dx.doi.org/10.1039/c4ob02096k

Iskander G; Wood K; Eiffe E; Yee EMH; Black DS; Kumar N, 2015, 'ChemInform Abstract: Ritter Reactions of Isoflavanols: A Facile Route to 4‐Amidoisoflavans.', ChemInform, 46, http://dx.doi.org/10.1002/chin.201530197

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